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Authors whose works are in public domain in at least one jurisdiction

List of works by Kjetil Wessel Andressen

1-20 of 20 results

The serotonin 5-HT7 receptors: two decades of research

scientific article

Substrate specificities of g protein-coupled receptor kinase-2 and -3 at cardiac myocyte receptors provide basis for distinct roles in regulation of myocardial function

scientific journal article

Disheveled regulates precoupling of heterotrimeric G proteins to Frizzled 6.

scientific article published on 5 February 2014

Heterologous desensitization is evoked by both agonist and antagonist stimulation of the human 5-HT(7) serotonin receptor.

scientific article published on 17 February 2006

Activation of adenylyl cyclase by endogenous G(s)-coupled receptors in human embryonic kidney 293 cells is attenuated by 5-HT(7) receptor expression.

scientific article published on 27 September 2005

The inotropic effect of the active metabolite of levosimendan, OR-1896, is mediated through inhibition of PDE3 in rat ventricular myocardium

scientific article published on 4 March 2015

Synthesis and in vitro evaluation of small-molecule [18F] labeled gonadotropin-releasing hormone (GnRH) receptor antagonists as potential PET imaging agents for GnRH receptor expression.

scientific article

Identification of essential residues for binding and activation in the human 5-HT7(a) serotonin receptor by molecular modeling and site-directed mutagenesis

scientific article published on 8 May 2015

The atypical antipsychotics clozapine and olanzapine promote down-regulation and display functional selectivity at human 5-HT7 receptors.

scientific article published on 12 June 2015

Brain penetrant small molecule (18)F-GnRH receptor (GnRH-R) antagonists: Synthesis and preliminary positron emission tomography imaging in rats.

scientific article

Biochemical and pharmacological study of N‐linked glycosylation of the human serotonin 5‐HT7(a) receptor

scientific article published on April 25, 2012

Acidic biphenyl derivatives: synthesis and biological activity of a new series of potent 5-HT(4) receptor antagonists

scientific article published on 11 September 2013

Synthesis and pharmacological properties of a new hydrophilic and orally bioavailable 5-HT4 antagonist

scientific article published on April 9, 2013

Related GPCRs couple differently to Gs: preassociation between G protein and 5-HT7 serotonin receptor reveals movement of Gαs upon receptor activation.

scientific article published on 27 October 2017

FRET-based cyclic GMP biosensors measure low cGMP concentrations in cardiomyocytes and neurons

scientific article published on 29 October 2019

An inactive receptor-G protein complex maintains the dynamic range of agonist-induced signaling

scientific article published on 16 November 2020

Preassociation between the 5-HT7 serotonin receptor and G protein Gs: molecular determinants and association with low potency activation of adenylyl cyclase

scientific article published on 03 December 2018

Construction of novel cGMP FRET-sensors based on PKG from Plasmodium falciparum.

scientific article published on 2 September 2015

Discovery and pharmacological profile of new hydrophilic 5-HT(4) receptor antagonists.

scientific article published on 5 July 2014

The 5-HT₇ serotonin receptor : G protein preassociation and functional selectivity

dissertation