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Optimisation of a triazolopyridine based histone demethylase inhibitor yields a potent and selective KDM2A (FBXL11) inhibitor

scientific article published in December 2014

Author/s

author: Christopher J. Schofield, Tobias Krojer, Frank von Delft, Akane Kawamura, Paul E. Brennan

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Work details

Publication date
December 1, 2014
- -
Language
English

Copyright status